GO 6976, also known as PD-406976, is a potent inhibitor of neurotrophin-receptor intrinsic tyrosine kinase. Gö 6976 blocked neurotrophin-induced signaling and autophosphorylation of neurotrophin-specific tyrosine kinase (Trk) receptors, either Trk B in cortical neurons or Trk A in GT1-1-trk9 cells.
中文名称:
12-(2-氰乙基)-6,7,12,13-四氢-13-甲基-5-氧代- 5H-吲哚并[2,3-a]吡咯并[3,4-c]咔唑
物化属性:
外观与形状:灰白色至黄色固体
密度:1.41
沸点:652.3ºC at 760 mmHg
折射率:1.773
闪光点:348.3ºC
PSA:62.75000
LOGP:4.92528